SJ-MX1830
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SKF-96365 hydrochloride
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SKF-96365 hydrochloride 是一种有效的 TRP channel 阻滞剂和 SOCE (store-operated Ca2+ entry) 抑制剂。SKF-96365 hydrochloride 可显著抑制豚鼠离体心脏 hERG、hKCNQ1/hKCNE1、hKir2.1 和 hKv4.3 电流,显著延长 QTc 间期。SKF-96365 hydrochloride 通过诱导结直肠癌细胞的细胞周期阻滞和凋亡 (apoptosis) 而显示出强大的抗肿瘤活性。
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SJ-MN0298
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Tanshinone IIA sulfonate sodium
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丹参酮IIA磺酸盐 |
Tanshinone IIA sulfonate sodium 是 tanshinone IIA 的衍生物,为 SOCE 的抑制剂,用于心血管疾病的研究。
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SJ-MX3853
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YM-58483
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YM 58483 (BTP2) is a SOCE blocker. SOCE has been found in macrophages, basophils, dendritic cells, and mast cells as well as T cells. YM 58483 has been reported to inhibit cytokine production and proliferation in T cells, and may serve as a potential medicinal candidate for treatment of bronchial asthma.
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SJ-MX2211
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Zegocractin (CM-4620)
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Zegocractin (CM-4620) 是一种钙离子释放激活通道 (CRAC channel) 的抑制剂,其对 Orai1/STIM1 和 Orai2/STIM1 的 IC50 值分别为 119 nM 和 895 nM。
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SJ-MX5724
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Synta66
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