货号 | 产品名 | 中文名称 | 产品描述 |
---|---|---|---|
SJ-MX3637 | ELN-441958 | ELN-441958 (ELN441958) is a novel, potent, and neutral bradykinin B1 Receptor antagonist which inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM. | |
SJ-BP0076A | Icatibant acetate | Icatibant acetate is a potent and specific synthetic peptide antagonist of bradykinin B2 receptor with an IC50 and Ki of 1.07 nM and 0.798 nM respectively. It inhibits bradykinin-induced contractions in isolated guinea pig ileum and pulmonary arteries as well as in rat uterus (IC50s = 11, 5.4, and 4.9 nM, respectively). | |
SJ-BP0291 | Bradykinin (1-5) | ||
SJ-BP0076 | Icatibant | 艾替班特 |
Icatibant 是有效的,特异的缓激肽B2受体拮抗剂,IC50 和 Ki 值分别为 1.07 nM 和 0.798 nM。 |
SJ-BP0262 | Bradykinin | 缓激肽 |
Bradykinin 是人体内的激肽物质,是由激肽释放酶-激肽系统产生的活性肽。Bradykinin 对 B2R 的选择性比 B1R 强10000 倍以上。Bradykinin 是炎症调节因子,也被认为是几种血管和肾功能以及神经调节因子。 |