SJ-MX2888
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Tetrabenazine Racemate
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丁苯那嗪外消旋体 |
Tetrabenazine Racemate is a selective and reversible inhibitor of vesicular monoamine transporter-2 (VMAT-2).
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SJ-MX2895
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Valbenazine
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Valbenazine is an inhibitor of vesicular monoamine transporter 2 (VMAT2). VMAT2 plays an important role in the packaging of monoamines into presynaptic vesicles. Valbenazine shows Ki values of 110 and 150 nM in rat striatum homogenates and human platelets, respectively. It is selective for VMAT2 over serotonin (5-HT) receptor subtypes 5-HT1A, 5-HT2A, and 5-HT2B and dopamine D1 and D2 receptors. It is used for the treatment of tardive dyskinesia.
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SJ-MX2726
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Tetrabenazine
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丁苯那嗪 |
Tetrabenazine (Ro 1-9569; trade name: Nitoman and Xenazin), a VMAT-inhibitor, is a drug for the treatment of symptomatic treatment of hyperkinetic movement disorder.
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SJ-MN0610
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Reserpine
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利血平 |
Reserpine 是囊泡单胺转运蛋白 2 (VMAT2) 的抑制剂。
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SJ-MN0610A
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Reserpine hydrochloride
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利血平盐酸盐 |
Reserpine hydrochloride是囊泡单胺转运蛋白 2 (VMAT2) 的抑制剂。
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SJ-MX2946
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(+)-Tetrabenazine
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(+)-丁苯那嗪 |
(+)-Tetrabenazine ((+)-TBZ; (3R,11bR)-TBZ; (3R,11bR)-Tetrabenazine) is a potent and reversible inhibitor of vesicular monoamine transporter 2 (VMAT-2) which inhibits transport by VMAT2 with 10-fold greater potency than transport by VMAT1.
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