货号 | 产品名 | 中文名称 | 产品描述 |
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SJ-MX3539 | 7ACC2 | 7ACC2 is a potent MCT inhibitor. Monocarboxylate transporters (MCTs) catalyze the proton-linked transport of monocarboxylates such as L-lactate, pyruvate, and the ketone bodies across the plasma membrane. There are four isoforms, MCTs 1-4, which are known to perform this function in mammals, each with distinct substrate and inhibitor affinities. | |
SJ-MX1650 | AR-C155858 | AR-C155858是选择性的单羧酸转运蛋白 MCT1 和 MCT2 抑制剂,Ki 分别为2.3 nM和10 nM。 | |
SJ-MX2729 | 7ACC1 | 香豆素D1421 | 7ACC1(DEAC; Coumarin D 1421; D 1421) selectively interfere with lactate fluxes in the lactate-rich tumor microenvironment; inhibits lactate influx but not efflux in tumor cells expressing MCT1 and MCT4 transporters. |
SJ-MX0111 | AZD3965 |
AZD3965是一种有效的选择性monocarboxylate transporter 1 (MCT1)抑制剂,结合亲和力为 1.6 nM; 它的选择性是 MCT2 的 6 倍。 |
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SJ-MX0952 | BAY-8002 | BAY-8002 是一种有效、选择性、可口服的单羧酸转运蛋白第 1 亚型 (monocarboxylate transporter 1 (MCT1)) 抑制剂,在表达 MCT1 的 DLD-1 细胞中,IC50 值为 85 nM,对 MCT1 的选择性远高于 MCT4。具有抗肿瘤活性。 | |
SJ-MX4059 | VB124 |
VB124 是一种有效的选择性 MCT4 抑制剂,特异性抑制表达 MCT4 的 MDA-MB-231 细胞的乳酸流出/输入,可用于心肌肥厚、心力衰竭和代谢的研究。 |
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SJ-MX5612 | α-cyano-4-hydroxycinnamic acid(α-CHCA) | α-氰基-4-羟基肉桂酸 |