货号 | 产品名 | 中文名称 | 产品描述 |
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SJ-MX0786 | MK-8245 |
MK-8245是一种有效的,靶向作用于肝脏的硬脂酰辅酶A去饱和酶(stearoyl-CoA desaturase,SCD)抑制剂,作用于人类SCD1时,IC50为1 nM,作用于大鼠和小鼠SCD1时,IC50为3 nM,具有抗糖尿病和抗高脂血症作用。 |
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SJ-MX2800 | A939572 | A939572 is a cell-permeable, potent and selective inhibitor of SCD1(stearoyl-CoA desaturase 1) (In vitro: IC50 = 37 nM for hSCD1, <4 nM for mSCD1). Also exhibited in vivo efficacy with dose-dependent desaturation index lowering effect. SCD1 inhibition resulted in alterations in macrophage membrane lipid composition and marked hypersensitivity to toll-like receptor 4 agonists. | |
SJ-MX2462 | MF-438 | MF-438 是一种有效且口服生物可利用的 stearoyl-CoA desaturase 1 (SCD1) 的抑制剂,对 rSCD1 的 EC50 值为 2.3 nM。 | |
SJ-MX1284 | O-Phospho- L-serine | PluriSIn 1 (NSC 14613) 是一种酰基-辅酶A去饱和酶 (SCD) 抑制剂,是一种多能细胞特异性的抑制剂。 |