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Bradykinin Receptor

Bradykinin Receptor相关产品(5)
货号 产品名 中文名称 产品描述
SJ-MX3637 ELN-441958 ELN-441958 (ELN441958) is a novel, potent, and neutral bradykinin B1 Receptor antagonist which inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.
SJ-MX3744 SSR240612 SSR-240612 is a potent and selective, non-peptide antagonist of the bradykinin B1 receptor (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors, respectively). It inhibits the contraction of rabbit aorta and rat ileum induced by the B1 receptor agonist des-Arg9-bradykinin (des-Arg9-BK) ex vivo in a concentration-dependent manner.
SJ-BP0076 Icatibant 艾替班特

Icatibant 是有效的,特异的缓激肽B2受体拮抗剂,IC50 和 Ki 值分别为 1.07 nM 和 0.798 nM。

SJ-BP0262 Bradykinin 缓激肽 Bradykinin是由激肽释放酶-激肽系统产生的活性肽。 它是炎症调节因子,也被认为是几种血管和肾功能以及神经调节因子。
SJ-BP0076A Icatibant acetate Icatibant acetate is a potent and specific synthetic peptide antagonist of bradykinin B2 receptor with an IC50 and Ki of 1.07 nM and 0.798 nM respectively. It inhibits bradykinin-induced contractions in isolated guinea pig ileum and pulmonary arteries as well as in rat uterus (IC50s = 11, 5.4, and 4.9 nM, respectively).