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Glucocorticoid Receptor

Glucocorticoid Receptor相关产品(50)
货号 产品名 中文名称 产品描述
SJ-MX3713 Velsecorat

Velsecorat (AZD7594, AZ13189620) 是一种有效的,选择性非甾体类糖皮质激素受体 (glucocorticoid receptor) 调节剂,IC50 值为 0.9 nM。

SJ-MH0019B Prednisolone disodium phosphate 泼尼松龙21-磷酸二钠 Prednisolone sodium phosphate is a water soluble form of prednisolone and a glucocorticoid with anti-inflammatory and immunomodulating properties. It is used to treat a variety of inflammatory and autoimmune conditions and some cancers. It is the active metabolite of the drug prednisone and is used especially in patients with liver failure, as these individuals are unable to metabolize prednisone into active prednisolone.
SJ-MH0032 Flunisolide 氟尼缩松 Flunisolide is a synthetic corticosteroid with anti-inflammatory and antiallergic properties.
SJ-MH0040 Betamethasone dipropionate 二丙酸倍他米松 Betamethasone dipropionate (Alphatrex; BetaVal; Diprolene; SCH-11460; SCH11460; Diprolene AF; Diprosone; Luxiq; Betamethasone 17,21-dipropionate) is a synthetic glucocorticoid steroid with anti-inflammatory and immunosuppressive activities. It is approved as a topical cream, ointment, lotion or gel (Diprolene) to treat itching and other minor skin conditions such as eczema.
SJ-MH0041 Betamethasone valerate Betamethasone Valerate (BV; BET; Betoid; Valison; 9α-Fluo; Valisone; Bedermin; Betneval; Beta-Val; Bextasol; Dermosol; Stanoval) is a moderately potent and commonly used glucocorticoid steroid with anti-inflammatory and immunosuppressive activities. Betamethasone valerate is approved as an anti-inflammatory corticosteroid for topical applications.
SJ-MX2479 Beclometasone dipropionate 二丙酸倍氯米松

Beclometasone dipropionate 是 Beclometasone 的前体药物,是口服有效的糖皮质激素受体激动剂。Beclometasone dipropionate 通过糖皮质激素受体发挥作用,抑制炎症和过度增殖。Beclometasone dipropionate 可用于哮喘研究。

SJ-MX2922 Mometasone furoate 糠酸莫米松 Mometasone furoate (Sch32088) 是一种糖皮质激素受体 (glucocorticoid receptor) 激动剂,具有抗炎和抗过敏活性。Mometasone furoate 作为皮质类固醇类试剂,动物模型中,用于慢性皮肤湿疹和气道炎症以及哮喘的局部应用。
SJ-MH0064 Methylprednisolone acetate Methylprednisolone acetate is a novel and potent glucocorticoid.
SJ-MH0068 Desonide Desonide is a low-potency topical corticosteroid.
SJ-MH0072 Loteprednol Etabonate Loteprednol Etabonate is an anti-inflammatory corticosteroid used in optometry and ophthalmology.
SJ-MH0077 Fluocinonide 氟轻松 Fluocinonide is a potent glucocorticoid/corticosteroid that has been approved for use as a topical anti-inflammatory drug for the treatment of skin disorders such as seborrhoeic dermatitis and eczema.
SJ-MH0080 Deflazacort 地夫可特 Deflazacort (ML-458; ML458; DL-458-IT, L-5458) is a potent glucocorticoid drug approved for use as an anti-inflammatory and immunosuppressant.
SJ-MH0081 Triamcinolone 曲安西龙 Triamcinolone (BRN2341955), a long-acting synthetic corticosteroid, is an approved glucocorticoid medication with anti-inflammatory activities. Itcan be applied topically for the management of various disorders such as eczema, psoriasis, arthritis, allergies, ulcerative colitis, lupus, etc.
SJ-MH0082 Meprednisone 泼尼松 Meprednisone is a glucocorticoid and a methylated derivative of prednisone.
SJ-MH0015 Ciclesonide 环索奈德 Ciclesonide (RPR251526) 是一种具有强效抗炎活性的糖皮质激素,可用于哮喘研究。
SJ-MX2124 AL 082D06 AL 082D06 是一种选择性的非甾体类糖皮质激素受体 (GR) 拮抗剂,Ki 为 210 nM。
SJ-MH0024A Hydrocortisone Acetate 醋酸氢化可的松 Hydrocortisoneacetate是一种皮质类固醇,用来减少轻微皮肤刺激或痔疮引起的肿胀,搔痒和疼痛。
SJ-MH0012 Fluticasone propionate 丙酸氟替卡松 Fluticasone propionate 是一种有效的局部抗炎激素,一种选择性的糖皮质激素受体 (glucocorticoid receptor) 激动剂,绝对亲和力 KD 为 0.5 nM。Fluticasone propionate 在其他甾体受体上几乎没有活性。具有抗病毒活性。
SJ-MX5641 AZD9567 AZD9567 (compound 15) 是一种有效的、具有口服活性的、非甾体类的、选择性糖皮质激素受体调节剂 (SGRM), 其 IC50 值为 3.8 nM。对 SCW 联合炎症表现出良好的疗效。
SJ-MX5727 Mapracorat Mapracorat 是新型的非甾类有选择性的 glucocorticoid receptor 激动剂。